Bioactive Small Molecules
Cayman Chemical SU 4942, Purity: ≥98%, CAS: 76086-99-2, 100 mg
A modulator of tyrosine kinase signaling; inhibits VEGF- or acidic FGF-induced mitogenesis of endothelial cells in vitro
Medchemexpress LLC HY-19024 5mg Medchemexpress, Merbarone CAS:97534-21-9 Purity:>98%
Medchemexpress, HY-19024 5mg Merbarone CAS:97534-21-9 Merbarone (NSC 336628) is an orally active inhibitor of topoisomerase II. Merbarone acts primarily by blocking topoisomerase II-mediated DNA cleavage without stabilizing topo II-DNA covalent complexes. Merbarone is an anticancer agent[4]. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Cayman Chemical SEN-12333, Purity: ≥98%, CAS: 874450-44-9, 100 mg
An agonist of α7 nAChRs (Ki = 0.26 µM); selective for α7 nAChRs over α1-, α3-, and α4β2 subunit-containing nAChRs and the 5-HT3 receptor, as well as a panel of 70 additional neurotransmitter, growth factor, and peptide receptors at 10 µM; activates the α7 nAChR in GH4C1 cells expressing the rat receptor (EC50 = 1.6 µM); topical application prevents decreases in the number of retinal ganglion cells in a rat model of glaucoma; reverses scopolamine- or MK-801-induced memory deficits in the novel objection recognition test in rats at 3 mg/kg
TARGETMOL CHEMICALS INC PKI-402 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg and bulk. Please contact Fisher for quotes. PKI-402 is a potent PI3K and mTOR inhibitor. PKI-402 inhibits PI3K(alpha) mTOR PI3K(beta) PI3K(delta) and PI3K(gamma) with IC50s of 2 3 7 14 and 16 nM respectively. purity: 100%
Medchemexpress LLC HY-113407A 50mg Medchemexpress, D-Fructose-6-phosphate (disodium) salt CAS:26177-86-6 Purity:>98%
Medchemexpress, HY-113407A 50mg D-Fructose-6-phosphate (disodium) salt CAS:26177-86-6 D-Fructose-6-phosphate disodium salt is an endogenous metabolite. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Apexbio Technology LLC Protease Inhibitor Cocktail (100X in DMSO, EDTA plus), 20x(1ml A + 1ml B)
Protease Inhibitor Cocktail (100X in DMSO, EDTA plus), which is used during cell lysis and protein extraction, is a ready-to-use concentrated stock solutions of multiple protease inhibitors for endogenous protease. This product contains a separate 0.5M EDTA solution which inhibiting metalloproteases. It generates optimized concentrations of six broad-spectrum protease inhibitors stabilized in DMSO, that powerfully inhibits serine-proteases, cysteine-proteases, aspartic acid-proteases and aminopeptidases appearing in cellular lysate samples. EDTA provides inhibition for metalloproteases. Other sizes are available. Please inqury us for quote.
Medchemexpress LLC HY-111406 5mg Medchemexpress, Omidenepag isopropyl CAS:1187451-19-9 Purity:>98%
Medchemexpress, HY-111406 5mg Omidenepag isopropyl CAS:1187451-19-9 Omidenepag isopropyl is a selective EP2 receptor agonist. Omidenepag isopropyl is converted to the active product Omidenepag during corneal penetration, and Omidenepag is a highly selective EP2 receptor agonist. Omidenepag isopropyl shows only weak affinity for EP1, EP2, and FP receptors. Omidenepag isopropyl is under development for the treatment of glaucoma as an intraocular pressure (IOP)-lowering drug. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
TARGETMOL CHEMICALS INC DZ2002 5MG
Also available in 1 mg 2 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. DZ2002 is an orally active reversible and low-cytotoxic type III SAHH inhibitor (Ki=17.9 nM) with good immunosuppressive activity. DZ2002 prevents the development of experimental dermal fibrosis by reversing the profibrotic phenotype of various cell types. DZ2002 can be used in studies of autoimmune diseases such as lupus syndrome and systemic sclerosis. purity: 98%
![eMolecules 25387-67-1 | Sodium Camptothecin | AA Blocks LLC388.355 | C20H17N2NaO5 | 0.000 | [Na+].CCC(O)(C([O-])=O)c1cc2-c3nc4ccccc4cc3Cn2c(=O)c1CO | 250mg | 795057185](https://assets.fishersci.com/TFS-Assets/CCG/product-images/NC3967272.jpg-250.jpg)
eMolecules 25387-67-1 | Sodium Camptothecin | AA Blocks LLC388.355 | C20H17N2NaO5 | 0.000 | [Na+].CCC(O)(C([O-])=O)c1cc2-c3nc4ccccc4cc3Cn2c(=O)c1CO | 250mg | 795057185
Sodium Camptothecin | AA Blocks LLC | 25387-67-1388.355 | C20H17N2NaO5 | 0.000 | [Na+].CCC(O)(C([O-])=O)c1cc2-c3nc4ccccc4cc3Cn2c(=O)c1CO | 250mg | 795057185
Medchemexpress LLC Stearoyl glutamic acid sodium | 38517-23-6 | C23H42NNaO5 | 1 G
Stearoyl glutamic acid sodium (Sodium stearoyl glutamate) is an anionic emulsifier and surfactant suitable for use in cosmetics. It also functions as an amino acid alkyl amide sensitizer and a chelating agent. While it may cause allergic contact dermatitis, it is noted for its emulsifying properties and preservative efficacy.
- Increases apparent viscosity in O/W emulsions.
- Reduces particle size in O/W emulsions.
- Enhances particle size uniformity in O/W emulsions.
- Improves long-term physical stability in O/W emulsions.
- Demonstrates excellent preservative efficacy in FB1 emulsion, eliminating tested bacteria, yeasts, and fungi within 7 days and maintaining microbial sterility for up to 28 days.
Medchemexpress LLC (R)-7-cyano-2,3,4,5-tetrahydro-1-(1H-imidazol-4-ylmethyl)-3-(phenylmethyl)-4-(2-thienylsulfonyl) | 195987-41-8 | 99.9% | 489.61 g/mol | C25H23N5O2S2 | 10 MG
A small-molecule farnesyl transferase inhibitor supplied as a high-purity solid for research use. It inhibits prenylation of Ras family proteins and is intended for laboratory studies requiring a selective FTase inhibitor.
- High purity (99.9%)
- Solid form, suitable for formulation or dissolution
- Molecular weight 489.61 g/mol
- Chemical formula C25H23N5O2S2
- Recommended storage: powder -20°C for long term; solvent storage guidelines available
- Available as a 10 mg research pack
![Medchemexpress LLC N-[[4-methyl-2-(2-thienyl)-5-thiazolyl]methyl]-N′-2-thienyl-urea | 1396814-79-1 | 98.5% | 335.47 g/mol | C14H13N3OS3 | 10 MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/5000288519.png-250.jpg)
Medchemexpress LLC N-[[4-methyl-2-(2-thienyl)-5-thiazolyl]methyl]-N′-2-thienyl-urea | 1396814-79-1 | 98.5% | 335.47 g/mol | C14H13N3OS3 | 10 MG
VU0542270 is a small-molecule research compound that selectively inhibits vascular Kir6.1/SUR2B ATP-sensitive potassium (KATP) channels and is used in cellular and biochemical assays to study SUR2B/Kir6.1-mediated KATP channel function. Reported potency is in the low-hundreds of nanomolar range, and the supplied sample is high-purity solid for laboratory research.
- Selective inhibitor of vascular Kir6.1/SUR2B KATP channels.
- Reported potency: IC50 ≈ 0.10-0.13 μM.
- High purity suitable for biochemical and cellular assays.
- Supplied as a 10 mg solid research sample.
- Commonly used in pharmacological and mechanistic studies of KATP channels.
Medchemexpress LLC 6-Amino-N-(2-(diethylamino)ethyl)quinoline-2-carboxamide | 1429047-67-5 | 99.7% | C16H22N4O | 100 MG
6-Amino-N-(2-(diethylamino)ethyl)quinoline-2-carboxamide is a chemical compound that serves as a drug intermediate for the synthesis of various active compounds. It is supplied as a solid with high purity.
- High purity: 99.7%
- Stable as powder at -20°C for 3 years, or 4°C for 2 years
- Soluble in DMSO at 100 mg/mL
- Used for the synthesis of active compounds
Medchemexpress LLC Depressine | 176182-06-2 | 1 MG
Depressine is an iridoid glycoside isolated from the methanol extract of the aerial parts of Gentiana depressa. It can be used to reduce oxidative DNA base damage and strand breaks that are prone to occur during the preparation of silver nanoparticles (AgNPs).
- Iridoid glycoside
- Isolated from Gentiana depressa
- Reduces oxidative DNA base damage
- Reduces strand breaks during silver nanoparticle preparation
- Molecular weight: 688.63
- Molecular formula: C30H40O18
- Appearance: solid, white to light yellow
- Purity: 99.84%
Medchemexpress LLC HY-W009362 50mg Medchemexpress, DL-Isocitric acid (trisodium salt) CAS:1637-73-6 Purity:>98%
Medchemexpress, HY-W009362 50mg DL-Isocitric acid (trisodium salt) CAS:1637-73-6 DL-Isocitric acid trisodium salt is an endogenous metabolite. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.